Coluracetam (135463-81-9) - Cofttek

Coluracetam (135463-81-9)

Bari 8, 2021

Cofttek shine mafi kyawun masana'antar foda ta Coluracetam a China. Masana'antarmu tana da cikakken tsarin sarrafa sarrafawa (ISO9001 & ISO14001), tare da damar samarwa kowane wata na 160kg.

 


Status:A cikin Mas Samar
Naúra:1kg / jaka, 25kg / Drum

Coluracetam (135463-81-9) Sfasali

name:Coluracetam
CAS:135463-81-9
tsarki98%
Formula kwayoyin:C19H23N3O3
Kwayoyin Weight:341.411 g / moll
Shawarwar Melt:N / A
Chemical name:N-(2,3-dimethyl-5,6,7,8-tetrahydrofuro[2,3-b]quinolin-4-yl)-2-(2-oxopyrrolidin-1-yl)acetamide

Saukewa: MKC-231

Bci-540

Kamancin:Coluracetam; BCI-540; MKC-231; BCI 540; MKC 231; BCI540; MKC231.
InChI Key:PSPGQHXMUKWNDI-UHFFFAOYSA-N
Rabin Rayuwa:N / A
Solubility:Soluble a DMSO
Yanayin Adana:Dry, duhu kuma a 0 - 4 C don gajere (kwanaki zuwa makonni) ko -20 C na dogon lokaci (watanni zuwa shekaru)
Aikace-aikace:raw Coluracetam foda (MKC-231) magani ne na racetam na roba wanda aka ɗauka ya zama fili na nootropic.
Appearance:Farin crystalline foda

 

Coluracetam (135463-81-9) NMR Spectrum

Coluracetam (135463-81-9) Bakan NMR

Idan kuna buƙatar COA, MSDS, HNMR don kowane samfurin samfur da sauran bayanai, da fatan za a tuntuɓi mu manajan talla.

 

Mene ne Coluracetam (135463-81-9)?

Raw Coluracetam foda (MKC-231) wani maganin racetam ne mai raɗaɗin ƙwayoyi wanda ake zaton ya zama wuri mai mahimmanci. Ba shi da babban shaidar shaida da ke binciken shi, amma tsarin aikin (da kuma tsari) ya kasance mai banbanci daga sauran mahallin magunguna irin su Piracetam ko Aniracetam.

Raw Coluracetam foda ya bayyana yana hulɗa tare da tsarin da aka sani da babban haɗin gwiwar choline (HACU a takaice), wanda shine matakin iyakacin iyaka na zana choline a cikin neuron don haɗuwa a cikin neurotransmitter acetylcholine. Haɓaka ƙimar HACU yana bayyana yana haɓaka ayyukan ƙwayoyin ƙwayoyin cuta na cholinergic, don haka manufa ce da ake so. haɓakar fahimi.

 

Coluracetam (135463-81-9) amfanin

  • Inganta ƙwaƙwalwar ajiya da Koyo
  • Inganta Karatun Karatu da kuma Karatatawa kyauta
  • Inganta Cigaban Lokaci
  • Rage Rashin Yin Jiyya-Juriya
  • M Neurogenesis ingantawa
  • Za a iya inganta Rashin Ilimin tunanin mutum
  • Zan Iya Inganta hangen nesa
  • Ciwo mara lafiya na Ciwon kwancen Ciwon kwankwasiyya
  • Amfani da nishaɗin Coluracetam

 

Coluracetam (135463-81-9) amfani

Coluracetam (INN) (lambar suna BCI-540; da MKC-231) foda shine wakili na nootropic na dangin racetam. Kamfanin Mitsubishi Tanabe Pharma ne ya kirkiro shi kuma ya gwada shi don cutar Alzheimer. Bayan da maganin ya gaza kaiwa ga ƙarshe a cikin gwaje-gwajensa na asibiti BrainCells Inc ya ba shi lasisi don yin bincike kan babbar matsalar rashin damuwa (MDD), wanda aka rigaya ta ba shi kyautar "Grangarwar Shirin Gano Maganin Cancanta" ta jihar California.

 

Coluracetam (135463-81-9) sashi

Yawancin bincike akan coluracetam an yi a kan dabbobi maimakon mutane, saboda haka babu wata takaddama ta hanyar yarda da duniya. Ana amfani dashi mai mahimmanci azaman kayan aiki kamar 5-20 MG. Masu amfani da coluracetam sun bayar da rahoto kan iyakokin maganin da ake gudanarwa a cikin layi da kuma a hankali.

Bayanin mai amfani kuma ya ambata cewa haƙuri ga coluracetam foda na iya haɓaka da sauri. Kamar yadda yake tare da dukkan magunguna, musamman nootropics, yana da kyau a fara a ƙananan allurai kuma a ƙara kashi a hankali yayin da jikinku yake amsawa kuma ya daidaita da magani. Coluracetam ba mai guba bane kuma ana ɗaukarsa mai juriya da aminci.

 

Coluracetam foda na siyarwa(Inda zaka Sayi Coluracetam foda a cikin girma)

Kamfaninmu yana jin daɗin dogon lokaci tare da abokan cinikinmu saboda muna mai da hankali kan abokin ciniki sabis da samar da manyan samfurori. Idan kuna sha'awar samfuranmu, muna da sassauƙa tare da tsara umarni don dacewa da takamaiman buƙatarku kuma lokacin saurin jagorancinmu akan umarni yana bada tabbacin za ku ɗanɗana samfurinmu akan lokaci. Har ila yau, muna mai da hankali kan ƙarin sabis ɗin ƙimar. Muna nan don tambayoyin sabis da bayani don tallafawa kasuwancin ku.

Mu masu sana'a ne na Coluracetam foda na shekaru masu yawa, muna samarwa samfurori tare da gasa farashin, kuma samfurin mu yana da inganci mafi girma kuma yana fuskantar ƙaƙƙarfan gwaji mai zaman kansa don tabbatar da cewa yana da aminci don amfani a duk duniya.

 

References

[1] Akaike A, et al. (1998). Tasirin kariya na MKC-231, ingantaccen dangantaka mai ɗauke da haɓaka, a kan yaduwar ƙwayar cuta a cikin ƙananan ƙwayoyin cuta. Jpn J Pharmacol.

[2] Bessho, T., Takashina, K., Tabata, R., Ohshima, C., Chaki, H., Yamabe, H., Egawa, M., Tobe, A., & Saito, K. (1996). Hanyoyin da ke tattare da haɓakar haɓakar haɓaka mai haɓaka 2- (2-oxopyrrolidin-1-yl) -N- (2,3-dimethyl-5,6,7,8-tetrahydrofuro [2,3-b] quinolin-4- yl) acetoamide akan karancin karatun koyon ruwa a beraye. Arzneimittel-Forschung, 46 (4), 369-373.

[3] Murai, S., Saito, H., Abe, E., Masuda, Y., Odashima, J., & Itoh, T. (1994). MKC-231, mai haɓaka haɓakar haɓaka, yana inganta ƙarancin ƙwaƙwalwar ajiyar ƙwaƙwalwar ajiya da rage haɓakar hippocampal acetylcholine da aka samu ta ion ethylcholine aziridinium ion a cikin beraye. Journal of Neural Transmission, 98 (1), 1-13. Doi: 10.1007 / bf01277590.

[4] Takashina K, Bessho T, Mori R, Eguchi J, Saito K. MKC-231, mai haɓaka haɓaka mai ƙarfi: (2) Tasiri akan haɗewar da sakin acetylcholine a cikin ratsan AF64A. J Canjin Jigilar Tsarin Kasa (Vienna). 2008 Jul; 115 (7): 1027-35. doi: 10.1007 / s00702-008-0048-1. PubMed PMID: 18446264.

[5] Shirayama Y, Yamamoto A, Nishimura T, Katayama S, Kawahara R. Sakamakon mai zuwa ga mai haɓaka mai haɓaka mai ƙarfi na MKC-231 yana haifar da ƙarancin halayen phencyclidine da raguwa a cikin ƙwayoyin septal cholinergic a cikin beraye. Eur Neuropsychopharmacol. 2007 Sep; 17 (9): 616-26. PubMed PMID: 17467960.

 


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