J-147 (1146963-51-0) - Cofttek

J-147 (1146963-51-0)

Bari 7, 2021

Cofttek shine mafi kyawun masana'antar foda J-147 a China. Masana'antarmu tana da cikakken tsarin sarrafa samarwa (ISO9001 & ISO14001), tare da damar samarwa kowane wata na 120kg.

 


Status:A cikin Mas Samar
Naúra:1kg / jaka, 25kg / Drum

J-147 (1146963-51-0) Sfasali

name:J-147
CAS:1146963-51-0
tsarki98%
Formula kwayoyin:C18H17F3N2O2
Kwayoyin Weight:350.341 g / mol
Shawarwar Melt:177-178 ° C
Chemical name:2,2,2-Trifluoroacetic acid 1-(2,4-Dimethylphenyl)-2-[(3-methoxyphenyl)methylene]hydrazide
Kamancin:N- (2,4-Dimethylphenyl) -2,2,2-trifluoro-N '- [(E) - (3-methoxyphenyl) methylene] acetohydrazide
InChI Key:HYMZAYGFKNNHDN-SSDVNMTOSA-N
Rabin Rayuwa:1.5 awo a cikin plasma da 2.5 hours a cikin kwakwalwa
Solubility:Matsaloli zuwa 100 mil a cikin DMSO kuma zuwa 100 mil a cikin ethano
Yanayin Adana:0 - 4 C don gajere (kwanaki zuwa makonni), ko -20 C na dogon lokaci (watanni)
Aikace-aikace:J-147 foda shine sabon gwaji maganin da ake haɓaka azaman magani mai yiwuwa don cutar Alzheimer.
Appearance:Farin farin-foda

 

J-147 (1146963-51-0) Bayanin NMR

J-147 (1146963-51-0)

Idan kuna buƙatar COA, MSDS, HNMR don kowane samfurin samfur da sauran bayanai, da fatan za a tuntuɓi mu manajan talla.

 

Menene J-147 (1146963-51-0)?

J-147 foda wani sabon magani ne na gwaji wanda aka haɓaka a matsayin yiwuwar maganin cutar Alzheimer. Ya zuwa yanzu, gwaje-gwajen da aka yi akan beraye suna nuna alƙawura da yawa. J147 ya ba da rahoton sakamako a cikin sake juyar da tasirin lalata da Alzheimer a cikin ƙirar linzamin kwamfuta. J147 daukan wani daban-daban m idan aka kwatanta da dama sauran Nootropics da Alzheimer ta kwayoyi. J147 yayi ƙoƙarin cire allunan adibas a cikin kwakwalwa. Masu bincike kuma sun lura cewa J147 yana da damar magance wasu batutuwan tsufa da yawa, ba kawai asarar ƙwaƙwalwar ajiya ba. Magungunan na iya taimakawa don hana zubar jini daga microvessels, kamar yadda aka nuna ta gwajin berayen da aka yi ya zuwa yanzu. An fara samar da maganin ne a cikin 2011. Tun daga wannan lokacin, an gudanar da gwaje-gwaje akan beraye amma ba mu ga wani faffadan gwajin asibiti na ɗan adam ba. Duk da haka, wasu bincike da aka buga a bara sun ba da hoto mai kyau na yadda J147 ke aiki a cikin kwakwalwar ɗan adam. A cewar takarda, maganin yana ɗaure da furotin mitochondria. Kwayoyin Mitochondria galibi suna da alhakin samar da makamashi. Ayyukan J147 akan su yana haɓaka farfadowar tantanin halitta. Wannan sabuntawa yana da mahimmanci a mayar da asarar ƙwaƙwalwar ajiya da haɓaka fahimi gabaɗaya kiwon lafiya.

 

J-147 (1146963-51-0) fa'idodi

Wataƙila Rashin Tsarin Digirin Digiri

J147 ya nuna alkawura da yawa a cikin jujjuyawar cututtukan ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwar ƙwaƙwalwa kamar Alzheimer da sauran su. A cikin gwaje-gwajen da aka yi a kan nau'ikan linzamin kwamfuta har zuwa yanzu, magungunan sun nuna matukar tasiri ga ma'amala da waɗannan yanayin.

J147 yana aiki ta hanyar taimaka wa sel a cikin kwakwalwa su sake farfadowa, yana sa su ƙarami kuma sun fi aiki fiye da tsofaffin ƙwayoyin. Koyaya, yana da mahimmanci a lura cewa ba a yi gwajin ɗan adam akan tasirin J147 ba. Da fatan hakan zai faru nan ba da jimawa ba amma har yanzu akwai magunguna don siyarwa azaman foda a cikin zaɓaɓɓun dillalai na kan layi.

 

Inganta Mitochondria Action da Longevity

J147 yana aiki ta hanyar ɗaure cikin mitochondria, ƙwayoyin da ke da alhakin samar da makamashi a jikinmu. Ayyukan J147 yana taimakawa wajen hana damuwa oxidative a cikin ƙwayoyin mitochondria, yana haifar da mafi kyawun aikin sel da tsawon rai.

J147 kuma yana taimakawa rage metabolites mai guba wanda zai iya haifar da wucewar ƙwayar cuta, tsari wanda sel ke mutuwa ta hanyar yin kwalliya sosai. Wannan yana ba da damar ƙwayoyinku su kasance cikin sabo da lafiya tsawon lokaci. A zahiri, wasu hanyoyin da aka yi akan batutuwan dabba sun nuna cewa gudanarwar J147 akan kwariyen 'ya'yan itace sun tsawaita rayuwarsu ta hanyar 9.5 zuwa 12.8%.

 

Inganta ƙwaƙwalwar ajiya

J147 ya kuma nuna alkawura da yawa tsakanin ƙirar motsi na gwaji a haɓaka ƙwaƙwalwa. Magungunan har ila yau sun taimaka wajen juyar da gawuwar ƙwaƙwalwa a cikin mazannin gwaji yayin nazarin binciken.

Masu binciken sun yi imanin cewa ana iya yin amfani da waɗannan tasirin a cikin abubuwan mutum. Hakanan akwai wasu hujjoji da ke ba da shawara cewa za a iya bincika J147 a matsayin magani don yiwuwar ƙwaƙwalwar sarari.

 

Yana Kare Neurons kuma Yana Taimakawa Girmar kwakwalwa

J147 kuma yana da kaddarorin neuroprotective waɗanda ke hana aikin hada ƙarfi abu a cikin sel. Wannan yana taimakawa kare neurons daga lalacewa mai yiwuwa. J147 na iya kasancewa mai haifar da ci gaban kwakwalwa. J147 na iya inganta synaptic plasticity a cikin kwakwalwa, yana haifar da ci gaba.

 

J-147 (1146963-51-0) amfani?

Yana Inganta Haɓakawa

J-147 kari yana haɓaka sarari da ƙwaƙwalwar ajiya na dogon lokaci. Magungunan miyagun ƙwayoyi yana juyar da lahani a cikin tsofaffi waɗanda ke fama da rashin fahimta. J-147 na siyarwa yana samuwa azaman adadin kan-da-counter kuma samari suna ɗauka don haɓaka ƙarfin koyo. Saukewa: J-147 anti-tsufa da kwayoyi Hakanan zai haɓaka ƙwaƙwalwar ajiya, hangen nesa, da tsabtar tunani.

 

Gudanar da Cutar Alzheimer

J-147 yana amfanar da marasa lafiya da cutar Alzheimer ta hanyar rage ci gaban yanayin. Misali, shan kari yana rage matakan beta-amyloid (Aβ) mai narkewa, wanda ke haifar da rashin aiki. Bayan haka, J-147 curcumin yana canza siginar neurotrophin don tabbatar da rayuwar neuronal, sabili da haka, ƙirƙirar ƙwaƙwalwar ajiya da cognition.

Marasa lafiya tare da AD suna da ƙananan abubuwan neurotrophic. Koyaya, shan ƙarin J-147 na Alzheimer yana haɓaka duka NGF da BDNF. Waɗannan ƙananan ƙwayoyin cuta suna taimaka wa ƙwaƙwalwar ajiya, koyo, da ayyukan fahimi.

 

J-147 (1146963-51-0) sashi

Karatu daban-daban sunyi amfani da nau'ikan maganin daban akan beraye, amma ɗayan karatun da aka inganta shine ya baiwa beraye 10 mg / kg na nauyin jiki kowace rana. Wani binciken ya yi amfani da magungunan 1, 3 ko 9 mg / kg, kuma ya sami sakamako mai dogaro da kashi, tare da ɗimbin ɗimbin aiki da kyau.

Koyaya, fassara wannan zuwa ƙimar ɗan adam na buƙatar daidaitawa don yanayin farfajiyar jiki. Dangane da tsarin jujjuyawar da aka fi amfani da shi, adadin daidai-daidaiton ɗan adam ya kamata ya daidaita sashin linzamin da aka raba ta 12.3 – ko .81 MG da kilogiram na nauyin jiki kowace rana.

Wannan .36 MG na J147 a kowace laban nauyin jiki kowace rana. Wannan zai zama MG 36 a rana don mutum mai fam ɗari, 54 MG ga mutum fam 150, ko 72 MG ga mutum fam 200.

Koyaya, sauran karatun sun sami sakamako mai kyau daga ƙananan ƙananan ƙwayoyi, kuma an basu cewa J147 yana ƙaddamar da kwakwalwa, ba a bayyane yake ba cewa sashi zaiyi daidai bisa girman jiki.

Kamar wannan, ya kamata a duba waɗannan lambobin azaman iyakokin sama, kuma akwai kowane dalili da za a gaskata cewa 10 zuwa 20 MG a rana ya isa ya sami wani sakamako.

 

J-147 foda na siyarwa(Inda zaka sayi foda J-147 a cikin girma)

Kamfaninmu yana jin daɗin haɗin kai tare da abokan cinikinmu saboda mun mai da hankali kan sabis na abokin ciniki da samar da samfuran manyan kayayyaki. Idan kuna da sha'awar samfurinmu, muna jujjuya tare da ƙirƙirar umarni don dacewa da takamaiman buƙatunku da lokacin jagoranmu na sauri akan umarni wanda zai ba ku tabbacin ku ɗanɗano samfurinmu akan lokaci. Hakanan muna mai da hankali kan ayyukan ƙara ƙimar. Muna samuwa don tambayoyin sabis da bayani don tallafawa kasuwancin ku.

Mu masu sana'a ne na J-147 foda na shekaru masu yawa, muna samarwa samfurori tare da gasa farashin, kuma samfurin mu yana da inganci mafi girma kuma yana fuskantar ƙaƙƙarfan gwaji mai zaman kansa don tabbatar da cewa yana da aminci don amfani a duk duniya.

 

References

[1] “Gwajin gwajin da aka yi niyyar cutar Alzheimer ya nuna tasirin tsufa” (Sanarwar sanarwa). Cibiyar Salk. 12 Nuwamba 2015. An dawo da Nuwamba 13, 2015.

[2] Brian L. Wang (13 Nuwamba 2015). Gwaji maganin da aka yi niyya ga cutar Alzheimer yana nuna rigakafin tsufa illa a gwaje-gwajen dabbobi. nextbigfuture.com. An dawo da Nuwamba 16, 2015.

[3] Solomon B (Oktoba 2008). “Filamentous bacteriophage a matsayin sabon maganin warkewa don maganin cutar Alzheimer”. Jaridar Cutar Alzheimer. 15 (2): 193–8. PMID 18953108.

 


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